17(R)-resolvin D1 specifically inhibits transient receptor potential ion channel vanilloid 3 leading to peripheral antinociception

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119
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SCOPUS

133

초록

BACKGROUND AND PURPOSE Transient receptor potential ion channel vanilloid 3 (TRPV3) is expressed in skin keratinocytes and plays an important role in thermal and chemical nociceptions in the periphery. The presence of TRPV3 inhibitors would improve our understanding of TRPV3 function and help to develop receptor-specific analgesics. However, little is known about physiological substances that specifically inhibit TRPV3 activity. Here, we investigated whether 17(R)-resolvin D1 (17R-RvD1), a naturally occurring pro-resolving lipid specifically affects TRPV3 activity.

키워드

17(R)-resolvin D1TRPV3specific inhibitorpainkeratinocytesnociceptive behavioursinflammationRESOLVIN D1CAPSAICIN RECEPTORINFLAMMATORY HYPERALGESIAMECHANICAL HYPERALGESIANOCICEPTIVE NEURONSSENSORY NEURONSPAINACTIVATIONTRPV3BRADYKININ
제목
17(R)-resolvin D1 specifically inhibits transient receptor potential ion channel vanilloid 3 leading to peripheral antinociception
저자
Bang, S.Yoo, S.Yang, T. J.Cho, H.Hwang, S. W.
DOI
10.1111/j.1476-5381.2011.01568.x
발행일
2012-02
유형
Article
저널명
British Journal of Pharmacology
165
3
페이지
683 ~ 692