Glycyrrhetinic acid as a hepatocyte targeting unit for an anticancer drug delivery system with enhanced cell type selectivity

  • Singh, Hardev
  • Kim, Seo Jin
  • Kang, Dong Hoon
  • Kim, Hye-Ri
  • Sharma, Amit
  • ... Kim, Jong Seung
  • 외 2명
Citations

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31

초록

Herein, we report the potential of glycyrrhetinic acid (GA) as an active targeting ligand for hepatocellular carcinoma (HCC) for the development of diagnosis/therapy using small-molecule based approaches. Our preliminary results demonstrated that GA-conjugation to diagnostic/therapeutic counterparts significantly enhanced their HCC targeting ability and excellent therapeutic efficacy.

키워드

HEPATOCELLULAR-CARCINOMAIN-VIVOCANCER-THERAPYLIVER-CANCERCHEMOTHERAPYPRODRUGAGENTSTHERANOSTICSDOXORUBICINACTIVATION
제목
Glycyrrhetinic acid as a hepatocyte targeting unit for an anticancer drug delivery system with enhanced cell type selectivity
저자
Singh, HardevKim, Seo JinKang, Dong HoonKim, Hye-RiSharma, AmitKim, Won YoungKang, ChulhunKim, Jong Seung
DOI
10.1039/c8cc05175e
발행일
2018-11-11
유형
Article
저널명
Chemical Communications
54
87
페이지
12353 ~ 12356