New types of potential BNCT agents, o-carboranyl aminoalcohols

  • Lee, Chai-Ho
  • Jin, Guo Fan
  • Joung, Jung Gun
  • Lee, Jong-Dae
  • Ban, Hyun Seung
  • 외 3명
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초록

o-Carboranyl aminoalcohols were synthesized using a standard Mannich reaction, and were tested for their anticancer properties using an in vitro test for CT26 cancer cells. The polar periphery of the aminoalcohols benefited from the high boron uptake in CT26 cancer cells with low toxicity, indicating their potential as BNCT agents. (C) 2009 Elsevier Ltd. All rights reserved.

키워드

Low cytotoxicityWater solubilityBoron neutron capture therapyBoron accumulationo-Carboranylphenol derivativesNEUTRON-CAPTURE THERAPYMANNICH CONDENSATIONSDERIVATIVES
제목
New types of potential BNCT agents, o-carboranyl aminoalcohols
저자
Lee, Chai-HoJin, Guo FanJoung, Jung GunLee, Jong-DaeBan, Hyun SeungNakamura, HiroyukiCho, Jung-KeunKang, Sang Ook
DOI
10.1016/j.tetlet.2009.03.207
발행일
2009-06-17
유형
Article
저널명
Tetrahedron Letters
50
24
페이지
2960 ~ 2963