Nitric oxide inhibitory and cytotoxic secondary metabolites from Talaromyces sp. BHM8-7

  • Han, Jae Sang; 
  • Lee, Dahyeon; 
  • Kim, Jun Gu; 
  • Jang, Joon Su; 
  • Dang, Vu Quan; 
  • ... Lee, Dongho; 
  • 외 4명
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초록

Two previously undescribed sesquiterpenes (1 and 2), one meroterpenoid (3), and one cyclic peptide (4), together with four known metabolites (5-8) were isolated from Talaromyces sp. BHM8-7. Their structures were elucidated by comprehensive spectroscopic techniques, such as 1D and 2D NMR, HRESIMS, ECD calculations, and the advanced Marfey's method following acid hydrolysis. Among the isolates, compound 5 exhibited significant inhibitory activity against nitric oxide (NO) production in LPS-stimulated RAW 264.7 cells without observable cytotoxicity. In addition, compounds 1 and 5 displayed potent cytotoxic effects on both SK-OV-3 and HCT-8 cells.

키워드

Sesquiterpenes; Meroterpene; Cyclic peptide; Anti-inflammatory effect; Cytotoxicity; Talaromyces sp; MARINE ISOLATE; FUNGUS; MEROTERPENOIDS; SESQUITERPENE; VERMISTATIN
제목
Nitric oxide inhibitory and cytotoxic secondary metabolites from Talaromyces sp. BHM8-7
저자
Han, Jae Sang; Lee, Dahyeon; Kim, Jun Gu; Jang, Joon Su; Dang, Vu Quan; Kim, Woo Jin; Lee, Dongho; Lee, Mi Kyeong; Lee, Jin Woo; Hwang, Bang Yeon
DOI
10.1016/j.phytochem.2026.114840
발행일
2026-07
유형
Article
저널명
Phytochemistry
권
247