Binary Drug Reinforced First Small-Molecule-Based Prodrug for Synergistic Anticancer Effects

  • Jangili, Paramesh
  • Won, Miae
  • Kim, Seo Jin
  • Chun, Jieun
  • Shim, Inseob
  • ... Kim, Jong Seung
  • 외 2명
Citations

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초록

We developed a small-molecule-based binary drug delivery system (BDDS) with two anticancer drugs, SN-38 and 5'-DFUR. The drug release from the prodrug BDDS can be achieved upon its reaction with intracellular H2O2, overexpressed in cancer cells. The efficacy of BDDS was demonstrated by a comparative study along with that of a single drug conjugate (SDDS), bearing SN-38 alone.

키워드

binary drugSN-385'-DFURCOX-2synergistic effect
제목
Binary Drug Reinforced First Small-Molecule-Based Prodrug for Synergistic Anticancer Effects
저자
Jangili, ParameshWon, MiaeKim, Seo JinChun, JieunShim, InseobKang, ChulhunRen, Wen XiuKim, Jong Seung
DOI
10.1021/acsabm.9b00418
발행일
2019-08-19
유형
Article
저널명
ACS Applied Bio Materials
2
8
페이지
3532 ~ 3539