siRNA Conjugate Delivery Systems

  • Jeong, Ji Hoon
  • Mok, Hyejung
  • Oh, Yu-Kyoung
  • Park, Tae Gwan
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초록

Small interfering RNA (siRNA) has been chemically conjugated to a variety of bioactive molecules, lipids, polymers, peptides, and inorganic nanostructured materials to enhance their pharmacokinetic behavior, cellular uptake, target specificity, and safety. To efficiently deliver siRNAs to the target cells and tissues, many different siRNA bioconjugates were synthesized and characterized, and their gene silencing efficiencies were tested in vitro and in vivo. In this review, recent developments of siRNA bioconjugates are summarized.

키워드

POLYELECTROLYTE COMPLEX MICELLESCELL-PENETRATING PEPTIDESSMALL INTERFERING RNAPOLY(ETHYLENE GLYCOL)-SIRNA CONJUGATETAT-DEPENDENT TRANSACTIVATIONCATIONIC FUSOGENIC PEPTIDECULTURED-MAMMALIAN-CELLSINNATE IMMUNE-RESPONSETARGETING IN-VIVOINTRACELLULAR DELIVERY
제목
siRNA Conjugate Delivery Systems
저자
Jeong, Ji HoonMok, HyejungOh, Yu-KyoungPark, Tae Gwan
DOI
10.1021/bc800278e
발행일
2009-01
유형
Review
저널명
Bioconjugate Chemistry
20
1
페이지
5 ~ 14