Expedient synthesis of 4-O-methylhonokiol via Suzuki-Miyaura cross-coupling

  • Kwak, Jae-Hwan
  • Cho, Young Ae
  • Jang, Jae-Yong
  • Seo, Seung-Yong
  • Lee, Heesoon
  • ... Lee, Kiho
  • 외 4명
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초록

Concise and practical synthesis of 4-O-methylhonokiol was achieved in 34% overall yield. The key features of our synthesis include chemoselective ortho-mono bromination of phenol as well as biaryl formation via Suzuki-Miyaura cross-coupling, in which bromophenol was reacted with potassium aryltrifluoroborate using Pd(OAc)(2) and RuPhos under microwave conditions. (C) 2011 Elsevier Ltd. All rights reserved.

키워드

Neolignan4-O-MethylhonokiolSuzuki-Miyaura cross-couplingPotassium aryltrifluoroborateCONCISE SYNTHESISNEOLIGNANSACIDS
제목
Expedient synthesis of 4-O-methylhonokiol via Suzuki-Miyaura cross-coupling
저자
Kwak, Jae-HwanCho, Young AeJang, Jae-YongSeo, Seung-YongLee, HeesoonHong, Jin TaeHan, Sang-BaeLee, KihoKwak, Young-ShinJung, Jae-Kyung
DOI
10.1016/j.tet.2011.09.115
발행일
2011-12-02
유형
Article
저널명
Tetrahedron
67
48
페이지
9401 ~ 9404