A fluorescence off-on reporter for real time monitoring of gemcitabine delivery to the cancer cells

  • Bhuniya, Sankarprasad
  • Lee, Min Hee
  • Jeon, Hyun Mi
  • Han, Ji Hye
  • Lee, Jae Hong
  • ... Kim, Jong Seung
  • 외 3명
Citations

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80
Citations

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85

초록

We present the design, synthesis, optical properties and in vitro biological assessments of the theranostic prodrug 6 in which a near IR fluorophore is conjugated with a cancer cell-directing biotin unit; further it is linked with the anti-cancer drug gemcitabine via a self-immolative spacer, a disulfide bond. The prodrug 6 is able to monitor drug delivery and cellular imaging.

키워드

APPENDED NAPHTHALIMIDETARGETED DELIVERYDRUG-RELEASENANOPARTICLESPRODRUGAPOPTOSISTHERAPY
제목
A fluorescence off-on reporter for real time monitoring of gemcitabine delivery to the cancer cells
저자
Bhuniya, SankarprasadLee, Min HeeJeon, Hyun MiHan, Ji HyeLee, Jae HongPark, NayoungMaiti, SukhenduKang, ChulhunKim, Jong Seung
DOI
10.1039/c3cc42653j
발행일
2013
유형
Article
저널명
Chemical Communications
49
64
페이지
7141 ~ 7143