Inhibitors of nitric oxide production from Artemisia princeps

  • Li, D.
  • Han, X.H.
  • Hong, S.S.
  • Lee, C.
  • Lee, M.S.
  • ... Lee, D.
  • 외 2명
Citations

SCOPUS

7

초록

The chromatographic separation of a methanol extract of Artemisia princes led to the isolation of two sesquiterpene lactones, artecanin (1) and canin (2), together with a flavonoid, eupatilin (3). Their structures were determined by 1D, 2D-NMR and MS data analysis. All of the isolates were evaluated for their potential to inhibit the LPS-induced production of nitric oxide in murine macrophage RAW 264.7 cells. Compounds 1-3 inhibited nitric oxide production with IC50 values of 19.5, 20.4 and 25.1 μM, respectively.

키워드

Artemisia princepsCompositaeNitric oxide production inhibitorSesquiterpene lactonemass spectrometrymedicinal plantmousenonhumannuclear Overhauser effectproton nuclear magnetic resonancethin layer chromatographyartecanincanineupatilinflavanoidlipopolysaccharidemethanolnitric oxide synthase inhibitorsesquiterpene lactoneunclassified druganimal cellartemisia princepsarticlecarbon nuclear magnetic resonancedrug isolationdrug mechanismdrug structuredrug synthesisIC 50macrophage
제목
Inhibitors of nitric oxide production from Artemisia princeps
저자
Li, D.Han, X.H.Hong, S.S.Lee, C.Lee, M.S.Lee, D.Lee, M.K.Hwang, B.Y.
발행일
2010
유형
Article
저널명
Natural Product Sciences
16
3
페이지
143 ~ 147