De novo generation of peptide binders with desired properties by deep generative models reinforced through enrichment of focused sets for iterative fine-tuning

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초록

Recurrent neural networks underwent reinforcement procedures for de novo generation of peptide binders with desired properties. Docking and scoring of peptides from these models allowed enrichment of focused sets with validated sequences for iterative fine-tuning, leading to reinforcement of those models. They enabled de novo generation of peptide sequences with high binding affinity to the target and possibly additional properties.

키워드

Peptides; Binding Affinities; Fine Tuning; Generative Model; Neural-networks; Peptide Sequences; Property; Recurrent Neural Networks; Amino Acid Sequence; Animal Experiment; Animal Model; Article; Binding Affinity; Controlled Study; Drug Analysis; Generative Model; Mouse; Nonhuman; Recurrent Neural Network; Artificial Neural Network; Chemistry; Metabolism; Molecular Docking; Peptide; Protein Binding; Molecular Docking Simulation; Neural Networks, Computer; Peptides; Protein Binding; DESIGN; LIGAND
제목
De novo generation of peptide binders with desired properties by deep generative models reinforced through enrichment of focused sets for iterative fine-tuning
저자
Oh, Doogie; Kim, Jongseong; Park, Yongdoo
DOI
10.1039/d5cc02530c
발행일
2025-05-23
유형
Article; Early Access
저널명
Chemical Communications
권
61
호
52
페이지
9488 ~ 9491